Orforglipron 0.5mg x 25 tablets
Orforglipron (LY3502970) is a non-peptide small-molecule GLP-1 receptor agonist developed by Eli Lilly. Unlike peptide-based GLP-1 receptor agonists, it activates the receptor through a small-molecule binding mode distinct from peptide agonists. Supplied strictly for in-vitro research and laboratory use only. Not for human or animal use.
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- Free Priority shipping on US orders over $100
- Ships same day on orders before 2 PM MST
- Plain, secure packaging
- Certificates published per tested lot — see current coverage
Mechanism of Action
Orforglipron is a non-peptide small-molecule agonist of the glucagon-like peptide-1 (GLP-1) receptor. It activates the receptor through a small-molecule binding mode distinct from peptide agonists. It is a GLP-1-only agent, distinct from tirzepatide, a dual GIP/GLP-1 peptide.
Properties
CAS Number
2212020-52-3
Molecular Formula
C₄₈H₄₈F₂N₁₀O₅
Molecular Weight
882.97 Da
Storage
Store at room temperature in a cool, dry place. Protect from moisture.
Shipping & Delivery
- Same-day dispatch on orders placed before 2 PM MST (Arizona — no daylight saving).
- US shipping from $5. Free Priority on orders $100+ (before discounts).
- Plain, unmarked packaging — no branding or product names on the outside.
- Ships to all 50 states, DC, Puerto Rico & the U.S. Virgin Islands; tracking emailed on every order.
Quality & Testing
- No third-party certificate has been published for this compound yet.
- USA-based; dispatched from Phoenix, Arizona.
- Supplied strictly for in-vitro laboratory research — not for human use.
Certificates are published for each lot we have tested — see the 14 published so far.
Research Applications
References & Citations
(1)Structural basis for GLP-1 receptor activation by LY3502970, an orally active nonpeptide agonist
Kawai T, Sun B, Yoshino H, et al.
Research Use Only
This product is intended strictly for in-vitro research, educational, and laboratory use. Not for human consumption. The information provided is based on published research and does not constitute medical advice.